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Glucagon-like peptide-1 (GLP-1) is a natural hormone that plays a role in maintaining normal blood glucose levels.4
As a practitioner caring for type 2 diabetes patients, you may see many individuals that struggle with high blood glucose. This is, at least in part, due to an inadequate GLP-1 RA response.1-3, 5
Loss in beta-cell mass[12]
Loss in beta-cell mass[12]
Decrease in beta-cell function[10]
Højberg PV, Vilsbøll T, Rabøl R, et al.
Four weeks of near-normalisation of blood glucose improves the insulin response to glucagon-like peptide-1 and glucose-dependent insulinotropic polypeptide in patients with type 2 diabetes. Diabetologia. 2009;52:199-207.
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The influence of GLP-1 on glucose-stimulated insulin secretion: effects on beta-cell sensitivity in type 2 and nondiabetic subjects. Diabetes. 2003;52:380-386.
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Secretion of glucagon-like peptide-1 in patients with type 2 diabetes mellitus: systematic review and meta-analyses of clinical studies. Diabetologia. 2013;56:965-972.
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Glucose metabolism and regulation: beyond insulin and glucagon. Diabetes Spectrum. 2004;17:183-190.
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Drucker DJ.
Mechanisms of action and therapeutic application of glucagon-like peptide-1. Cell Metab. 2018;27:740-756.
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GLP-1 receptor expression in human tumors and human normal tissues: potential for in vivo targeting. J Nucl Med. 2007;48:736-743.
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Glucagon-like peptide-1 and the central/peripheral nervous system: crosstalk in diabetes. Trends Endocrinol Metab. 2017;28:88-103.
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Incretin hormones: their role in health and disease. Diabetes Obes Metab. 2018;20:5-21.
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From the triumvirate to the ominous octet: a new paradigm for the treatment of type 2 diabetes mellitus. Diabetes. 2009;58:773-795.
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Loss of incretin effect is a specific, important, and early characteristic of type 2 diabetes. Diabetes Care. 2011;34(suppl2):S251-S257.
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Impairment of GLP1-induced insulin secretion: role of genetic background, insulin resistance and hyperglycaemia. Diabetes Obes Metab. 2012;14(suppl 3):85-90.
Nauck MA, Meier JJ.
GIP and GLP-1: stepsiblings rather than monozygotic twins within the incretin family. Diabetes. 2019;68:897-900.
Simonson G, Cuddihy R, Reader D, Bergenstal R.
International diabetes center treatment of type 2 diabetes glucose algorithm. Diabetes Manage. 2011:1:175-189.